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Heart Failure Congress 2009 Presentation
01 Jun 2009

Targeting the cardiorenal syndrome: adenosine A1 antagonists 

Webcasts available

Marco Metra 

Marco Metra
Topics: Heart Failure (HF)
Session number: 993
Session title: New Drugs on the horizon II
Authors: Metra, Marco (Brescia, IT)

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Kidney dysfunction is a major prognostic variable in patients admitted for acute heart failure (AHF).
Adenosine, through its action on type 1 receptors, causes afferent glomerular arteriole constriction in response to increased sodium delivery, as after loop diuretics administration. Adenosine type 1 receptor antagonists are a new class of agents for the treatment of AHF and cardio-renal syndrome. These agents have been shown to improve renal blood flow and glomerular filtration rate in patients with AHF and fluid overload.
In a pilot study , the adenosine type 1 receptor antagonist rolofylline has improved symptoms and outcomes in 182 patients with AHF.

This hypothesis has now been tested in a large multicenter trial (PROTECT) in 2000 patients with AHF, fluid overload, mild to moderate renal dysfunction, and high BNP/ NT-proBNP levels whose results will be available by the end of this year.

Teaching objective of the lecture:

Show the pathophysiologic basis and current evidence of the effects of adenosine type 1 receptor antagonists on renal function, symptoms and outcomes in the patients with acute heart failure, renal dysfunction and fluid overload.

Take home messages:

  • Role of kidney dysfunction in the prognosis of patients with acute heart failure
  • Results with adenosine type 1 receptor antagonists in patients with acute heart failure
  • Ongoing trials with adenosine type 1 receptor antagonists in heart failure.


The content of this article reflects the personal opinion of the author/s and is not necessarily the official position of the European Society of Cardiology.